CVT-10216

Descriptions

Biochem/physiol Actions

CVT-10216 possesses unequivocal anxiolytic properties. It will not affect the suppression of locomotor activity by mCPP (m-chlorophenylpiperazine).

CVT-10216 is a selective reversible inhibitor of aldehyde dehydrogenase-2 (ALDH-2), thereby inhibiting dopamine synthesis. CVT-10216 is active in suppressing alcohol and cocaine use, and anxiety.

General description

CVT-10216 is a 5-HT2c agonist.

Packaging

5, 25 mg in glass bottle

Specifications

Colour	white to beige
Quality Level	100
InChI key	YYOOFJZTRCPVFD-UHFFFAOYSA-N
InChI	1S/C24H19NO7S/c1-33(29,30)25-18-7-5-16(6-8-18)21-14-32-22-12-19(9-10-20(22)23(21)26)31-13-15-3-2-4-17(11-15)24(27)28/h2-12,14,25H,13H2,1H3,(H,27,28)
Manufacturer	SIGMA-ALDRICH
Solubility	DMSO: 10 mg/mL, clear
Form	powder
Assay	≥98% (HPLC)