5-BDBD, >=98% (HPLC)
Biochem/physiol Actions
5-BDBD is a specific inhibitor of P2X4. The compound inhibits P2X4 currents in CHO cells with an IC50 of 500 nM.
In native tissues, 5-BDBD is considered as a beneficial antagonist to analyze the effect of P2X receptors (P2XRs) subtype P2X4R.
Features and Benefits
This compound is featured on the P2 Receptors: P2X Ion Channel Family page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.
Packaging
5, 25 mg in glass bottle
| Colour | white to beige |
|---|---|
| Quality Level | 100 |
| InChI key | NKYMVQPXXTZHSF-UHFFFAOYSA-N |
| InChI | 1S/C17H11BrN2O2/c18-11-5-3-4-10(8-11)15-17-16(20-14(21)9-19-15)12-6-1-2-7-13(12)22-17/h1-8H,9H2,(H,20,21) |
| Manufacturer | SIGMA-ALDRICH |
| Solubility | DMSO: 15 mg/mL (clear solution) |
| Form | powder |
| Assay | ≥98% (HPLC) |
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