MRS 2395, >=98% (HPLC), solid

Descriptions

Biochem/physiol Actions

Antagonist for P2Y₁₂ purinoceptor; inhibits ADP-induced aggregation in rat platelets and antagonizes ADP-induced inhibition of cAMP in rat and human platelets in the presence of PGE1 without affecting P2Y₁ receptor-induced PLC activity in transfected astrocytoma cells.

Packaging

5, 25 mg in glass bottle

Specifications

Colour	white
Quality Level	100
InChI key	NASABYJQIYJDID-UHFFFAOYSA-N
InChI	1S/C20H30ClN5O4/c1-19(2,3)16(27)29-9-12(10-30-17(28)20(4,5)6)8-26-11-23-13-14(22-7)24-18(21)25-15(13)26/h11-12H,8-10H2,1-7H3,(H,22,24,25)
Manufacturer	SIGMA-ALDRICH
Solubility	DMSO: >10 mg/mL, H2O: insoluble
Form	solid
Assay	≥98% (HPLC)